8. 11th Frontiers in Medicinal Chemistry
- Session 1
‧Catalytic C-H Vinylation and Rearrangement of 1,5- and 1,4-Dipolar Quinolines
‧Nutrient-Mimetic PARP Inhibitor Conjugates for Improved Intracellular Exposure
‧Photocatalytic Direct Aromatic C-H Amination Using Saccharin
‧Cyclic Boronic Ester-Mediated Diastereoselective Alkenylation and its Application to Enantioselective Syntesis of Hasubanan Alkaloids
‧Electrochemical synthesis of stapled peptides via tyrosine arylation
Session 2
‧A Strategy to Discover Novel PROTACs Targeting Undruggable Proteins
‧Spiro-Hydantoin Derivatives as ADAMTS4 Onhibitors for the Treatment of MASLD
‧Total synteses and structure revisions of Menominin A & B
‧Bio-orthogonal incorporation of glutarimide to introduce the chemical degron for targeted protein degradation
Session 3
‧CDI-Mediated Urea Bond Formation: A Practical Approach to Urea-Containing Peptides
‧Microwave-Assisted Synthesis of Pyrrole-Imidazole Polyamides as Sequence-Selective DNA-Binding Modalities for Therapeutic Applications
‧Catalytic Enantioselective Construction of Biaryls via Photoredox Catalysis
‧Design, Synthesisn and Biological Evaluation of Novel Rubicon-Rab7 Interaction Inhibitors
‧연구재단 전략과제 PROTAC Platform 소개
- 충북대 약학대학 2관 201호
- 2026-08-20
